BDBM140977 US11547697, Compound 471::US9682141, 471

SMILES Nc1nc2cc(ccc2o1)-c1ccc2ncc(C(=O)N3CCC(F)(F)C3)n2c1

InChI Key InChIKey=JESLYQOGRZYKIG-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 140977   

LigandPNGBDBM140977(US11547697, Compound 471 | US9682141, 471)
Affinity DataIC50: >1.00E+4nMT: 2°CAssay Description:Briefly, the assay is a time resolved FRET assay that indirectly measures PIP3 product formed by the activity of a PI3-K. The kinase reaction is perf...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM140977(US11547697, Compound 471 | US9682141, 471)
Affinity DataIC50: >1.00E+4nMAssay Description:An exemplary system is PI 3-Kinase (human) HTRF? Assay from Upstate. The assay can be carried out according to the procedures suggested by the manufa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent